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索凡替尼发展历程
索凡替尼发展历程
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所属报告:
和黄医药-港股公司深度报告:出海不止呋喹替尼呋喹替尼不止结直肠癌-231102(55页).pdf
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索凡替尼全球临床研究进展
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行业数据
2025-04-07
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索凡替尼临床管线进展(截至2024年7月)
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行业数据
2025-04-07
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索凡替尼临床试验进度(截至24.7.1更新)
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行业数据
2025-01-24
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索凡替尼销售额(百万美元)
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行业数据
2025-01-24
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索凡替尼神经内分泌瘤市占率持续提升(%)
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竞争格局
2025-01-24
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索凡替尼:治疗NET的主要3级及以上TRAE
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行业数据
2024-12-31
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索凡替尼vs竞品国内NET治疗领域市场占有率
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行业数据
2024-12-31
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索凡替尼NET适应症销售预测(国内)
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行业数据
2024-12-31
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索凡替尼在所有来源的低级别神经内分泌瘤(NET)中均为I级推荐
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其它
2024-06-17
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预计索凡替尼治疗神经内分泌肿瘤患者中国销售峰值近8亿元
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其它
2024-06-17
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索凡替尼(苏泰坦)市占率快速提升
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竞争格局
2024-06-17
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索凡替尼是中国唯一获批用于胰腺和非胰腺来源的神经内分泌瘤
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其它
2024-06-17
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索凡替尼销售(百万美金)和增速(%)
5qC55o2u5Zu+54mH5Lit55qE5pWw5o2u77yM5Lul5LiL5piv6KGo5qC85bGV56S677yaCgp8IOW5tOS7vSB8IOW4guWcuumUgOWUrumine+8iOeZvuS4h+e+juWFg++8iSB8IOWinumAn++8iCXvvIkgfAp8LS0tLS0tfC0tLS0tLS0tLS0tLS0tLS0tLS0tLS18LS0tLS0tLS0tLXwKfCAyMDIxIHwgMTEuNiAgICAgICAgICAgICAgICAgfCAgICAgICAgICB8CnwgMjAyMiB8IDMyLjMgICAgICAgICAgICAgICAgIHwgKzE3OCUgICAgfAp8IDIwMjMgfCA0My45ICAgICAgICAgICAgICAgICB8ICszNiXvvIgrNDMlIENFUu+8iSB8CgrotYTmlpnmnaXmupDvvJrlkozpu4TljLvoja/lrpjnvZHjgIHlm73kv6Hor4HliLjnu4/mtY7noJTnqbbmiYDmlbTnkIY=
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其它
2024-05-27
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索凡替尼在神经内分泌瘤国内市场的占有率达到16%
5qC55o2u5Zu+54mH5Lit55qE5L+h5oGv77yM5Lul5LiL5piv5pWw5o2u55qE6KGo5qC877yaCgp8IOexu+WIqyAgIHwg5Y2g5pyJ546HIHwKfC0tLS0tLS0tfC0tLS0tLS0tfAp8IOWlpeabsuiCvSB8IDQyJSAgICB8Cnwg57Si5Yeh5pu/5bC8IHwgMTYlICAgIHwKfCDoiJLlsLzmm7/lsLwgfCAxNCUgICAgfAp8IOS+nee7tOiOq+WPuCB8IDEwJSAgICB8Cnwg5YW25LuWICAgfCAxOCUgICAgfAoK6LWE5paZ5p2l5rqQ77ya5ZKM6buE5Yy76I2vMjAyMuW5tOW5tOaKpea8lOekuuadkOaWme+8jOi0oumAmuivgeWIuOeglOeptuaJgA==
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行业数据
2023-04-20
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索凡替尼正是基于上述机制及血管抑制通路开发的一款新型口服酪氨酸激酶抑制剂(TKI),一方面通过抑制血管内皮生长因子受体(VEGFR1/2/3)和成纤维细胞生长因子受体(FGFR1)来抑制肿瘤新生血管生成;另一方面通过抑制 CSF-1R,减少 M2 型 TAM,促进机体对肿瘤细胞的免疫应答,从而发挥抗血管生成和免疫调节的双重活性。在动物实验中,索凡替尼可呈剂量、时间依赖性抑制肺组织中 VEGFR2磷酸化,从而有效抑制血管生成。在多种临床前模型上,索凡替尼均能够显著降低肿瘤体积,具有广谱抗肿瘤活性,以及对肿瘤微环境的免疫调节作用。
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和黄医药-港股公司深度报告:出海不止呋喹替尼呋喹替尼不止结直肠癌-231102(55页).pdf
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