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全球DPP1抑制剂管线情况
全球DPP1抑制剂管线情况
行业数据
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所属报告:
海思科(002653)-A股公司研究报告:创新转型成效显著多款新药上市放量-250929(48页).pdf
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《KAT6抑制剂化合物、药物组合物及其制备方法和N-(6-((1H-pyrazol-1-yl)methyl)-4-metho
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行业数据
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图10、全球PD-(L)1抑制剂市场规模(十亿美元)
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图10.VMAT2抑制剂全球销售情况(亿美元)
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行业数据
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全球PCSK9抑制剂市场规模(亿美元)
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市场规模
2026-04-13
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中国PCSK9抑制剂市场规模(亿人民币)
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市场规模
2026-04-13
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相较于PD-(L)1抑制剂,PD-(L)1/VEGF双抗有极大替代和拓展空间
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行业数据
2026-03-31
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全球在研FXI/FXIa抑制剂的临床进展
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行业数据
2026-02-26
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FXI/FXIa抑制剂全球可触及患者数
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行业数据
2026-02-26
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图表11FDA获批KRASG12C抑制剂的全球销售额(百万美元)
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行业数据
2026-02-25
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图表19KRASG12D抑制剂竞争格局
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竞争格局
2026-02-25
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图3 mCRC中EGFR抑制剂的美国收入(2004-2017)
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行业数据
2026-02-13
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主要JAK抑制剂全球销售额
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行业数据
2026-01-30
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国内主要JAK抑制剂在研格局
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JAK抑制剂:国内样本医院销售额
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DPP1 抑制剂 Brensocatib 于 2025 年 8 月获批,海思科同靶点的 HSK31858 全球研究进度领先。Brensocatib 是一种口服的可逆 DPP1 小分子抑制剂,可通过抑制 DPP1 及对NSPs 的激活,从而减少支气管扩张症等炎症性疾病造成的损害。2024 年 5 月,Insmed 宣布 Brensocatib 针对非囊性纤维化支气管扩张症患者的 III 期临床研究获得积极顶线结果,达到主要终点。该项研究的疗效分析包括 1680 名成人患者和 41 名青少年患者。在主要终点方面,10mg 和 25mg 剂量的 Brensocatib 分别将患者的年化肺部症状恶化(PE)率降低 21.1%和 19.4%,统计学显著并具有临床意义。此外,两种剂量的 Brensocatib 还达到了多个次要终点。2025 年 8 月 12 日,Insmed 宣布 Brensocatib(商品名:Brinsupri)获FDA 批准上市,用于治疗 12 岁及以上儿童和成人非囊性纤维化支气管扩张症患者,标志着该疾病领域迎来首款靶向治疗药物。目前,全球进入临床 III 期及以上阶段的 DPP1 抑制剂管线主要有 3 款,分别为 Insmed 的 brensocatib、海思科的 HSK31858 以及 Boehringer ingelheim 的 BI 1291583。其中,在国内市场,Insmed 的 brensocatib 尚未申报临床试验;2025 年 5 月,Boehringer ingelheim 的 BI 1291583 获批临床,拟开发治疗支气管扩张症;比较来看,海思科 HSK31858 处于国内领先位置,有望成为国内首个用于治疗支气管扩张的药物。
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